Name: R-30490

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Type: small molecule

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Groups: experimental

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Indication: Not Available

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Accession Number: DB09179 ( DB09179)

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Description: R-30490 is an opioid analgesic related to the highly potent animal tranquilizer carfentanil, and with only slightly lower potency. It was first synthesised by a team of chemists at Janssen Pharmaceutica led by Paul Janssen, who were investigating the structure-activity relationships of the fentanyl family of drugs. R-30490 was found to be the most selective agonist for the mu opioid receptor out of all the fentanyl analogues tested, but it has never been introduced for medical use in humans, although the closely related drug sufentanil is widely used for analgesia and anesthesia during major surgery.

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Structure:

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Prescription Products: Not Available

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Generic Prescription Products: Not Available

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Over the Counter Products: Not Available

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International Brands

• No Brands

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Brand Names

• No Brands

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Brand Mixtures

Brand Name	Ingredients

Brand Name	Ingredients

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Categories

• No Category

Indication: Not Available

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Pharmacodynamics: Not Available

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Mechanism of action: Not Available

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Absorption: Not Available

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Volume of distribution: Not Available

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Protein binding: Not Available

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Metabolism: Not Available

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Route of elimination: Not Available

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Half life: Not Available

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Clearance: Not Available

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Toxicity: Not Available

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Affected organisms

• Not Available

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SNP Mediated Adverse Drug Reactions

• Not Available

Manufacturers:

• Not Available

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Packagers:

• Not Available

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Dosage forms

Form	Route	Strength

Form	Route	Strength

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Prices

Unit description	Cost	Unit

Unit description	Cost	Unit

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Patents

Country	Patent Number	Approved	Expires (estimated)

Drug Interactions

Drug	Interaction

Drug	Interaction

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Food Interactions:

• Not Available

Kingdom: Organic compounds

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Super Class: Not Available

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Class: Not Available

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Sub Class: Not Available

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Direct Parent: Not Available

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Alternative Parents:

• Amino acids and derivatives
• Anilides
• Aralkylamines
• Azacyclic compounds
• Carbonyl compounds
• Dialkyl ethers
• Hydrocarbon derivatives
• Organic oxides
• Phenethylamines
• Tertiary carboxylic acid amides
• Trialkylamines

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substituent:

• Amine
• Amino acid or derivatives
• Anilide
• Aralkylamine
• Aromatic heteromonocyclic compound
• Azacycle
• Benzenoid
• Carbonyl group
• Carboxamide group
• Carboxylic acid derivative
• Dialkyl ether
• Ether
• Fentanyl
• Hydrocarbon derivative
• Monocyclic benzene moiety
• Organic nitrogen compound
• Organic oxide
• Organic oxygen compound
• Organonitrogen compound
• Organooxygen compound
• Phenethylamine
• Tertiary aliphatic amine
• Tertiary amine
• Tertiary carboxylic acid amide

Synthesis Reference: Not Available

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General Reference: Not Available

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External Links:

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Resource	Link

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ATC Codes:

• Not Available

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AHFS Codes:

• Not Available

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MSDS: Download