Detail

R-30490

Description

Name: R-30490
Type: small molecule
Groups: experimental
Indication: Not Available
Accession Number: DB09179 ( DB09179)
Description: R-30490 is an opioid analgesic related to the highly potent animal tranquilizer carfentanil, and with only slightly lower potency. It was first synthesised by a team of chemists at Janssen Pharmaceutica led by Paul Janssen, who were investigating the structure-activity relationships of the fentanyl family of drugs. R-30490 was found to be the most selective agonist for the mu opioid receptor out of all the fentanyl analogues tested, but it has never been introduced for medical use in humans, although the closely related drug sufentanil is widely used for analgesia and anesthesia during major surgery.
Structure:
Prescription Products: Not Available
Generic Prescription Products: Not Available
Over the Counter Products: Not Available
International Brands
  • No Brands

Brand Names
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Brand Mixtures
Brand NameIngredients

Categories
  • No Category

Pharmacology

Indication: Not Available
Pharmacodynamics: Not Available
Mechanism of action: Not Available
Absorption: Not Available
Volume of distribution: Not Available
Protein binding: Not Available
Metabolism: Not Available
Route of elimination: Not Available
Half life: Not Available
Clearance: Not Available
Toxicity: Not Available
Affected organisms
  • Not Available

SNP Mediated Adverse Drug Reactions
  • Not Available

Pharmacoeconomics

Manufacturers:
  • Not Available

Packagers:
  • Not Available

Dosage forms
FormRouteStrength

Prices
Unit descriptionCostUnit

Patents
CountryPatent NumberApprovedExpires (estimated)

Interactions

Drug Interactions
DrugInteraction

Food Interactions:
  • Not Available

Taxonomy

Kingdom: Organic compounds
Super Class: Not Available
Class: Not Available
Sub Class: Not Available
Direct Parent: Not Available
Alternative Parents:
  • Amino acids and derivatives
  • Anilides
  • Aralkylamines
  • Azacyclic compounds
  • Carbonyl compounds
  • Dialkyl ethers
  • Hydrocarbon derivatives
  • Organic oxides
  • Phenethylamines
  • Tertiary carboxylic acid amides
  • Trialkylamines

substituent:
  • Amine
  • Amino acid or derivatives
  • Anilide
  • Aralkylamine
  • Aromatic heteromonocyclic compound
  • Azacycle
  • Benzenoid
  • Carbonyl group
  • Carboxamide group
  • Carboxylic acid derivative
  • Dialkyl ether
  • Ether
  • Fentanyl
  • Hydrocarbon derivative
  • Monocyclic benzene moiety
  • Organic nitrogen compound
  • Organic oxide
  • Organic oxygen compound
  • Organonitrogen compound
  • Organooxygen compound
  • Phenethylamine
  • Tertiary aliphatic amine
  • Tertiary amine
  • Tertiary carboxylic acid amide

References

Synthesis Reference: Not Available
General Reference: Not Available
External Links:
ResourceLink

ATC Codes:
  • Not Available

AHFS Codes:
  • Not Available

MSDS: Download
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